Home The Active Ingredient Matrix Angelica sinensis (Ligustilide)

Formulation Intelligence

Angelica sinensis (Ligustilide)

Accelerate your CDMO or DTC pipeline. Map the exact physiochemical constraints, bioavailability synergies, and optimal delivery mechanisms for Angelica sinensis (Ligustilide).

Angelica sinensis, standardized for the phthalide ligustilide, functions as a potent vasodilator and anti-inflammatory agent primarily utilized for modulating gynecological health and improving microcirculation via smooth muscle relaxation.

Verified Molecular Profiling (NIH PubChem)

PubChem CID

5362922

Molecular Weight

210.32 g/mol

XLogP3 (Lipophilicity)

2.7

IUPAC Name

N-[(Z)-(2-methylcyclohexylidene)amino]pentanamide

Pharmacokinetic Synergies & Enhancers

Proven Synergy Pairings

  • Ferulic Acid for enhanced antioxidant protection of vascular endothelium
  • Astragalus membranaceus for synergistic immunomodulation and hematopoietic support

Biological Formulation Enhancers

  • Piperine for inhibition of glucuronidation to increase systemic ligustilide bioavailability
  • Medium-Chain Triglycerides (MCTs) for improved lipophilic solubilization and lymphatic transport

Delivery System Constraints & Modeling

Every active compound behaves uniquely based on the physical matrix it is suspended in. Below are the known physical chemistry challenges for Angelica sinensis (Ligustilide) across standard consumer modalities.

💊 Standard Capsules

Ligustilide is highly prone to oxidative degradation and volatilization, requiring airtight packaging or nitrogen flushing to maintain potency in dry powder capsules.

🍬 Gummy & Pectin Formats

The characteristic pungent, celery-like odor and bitter profile of ligustilide present significant organoleptic challenges that require complex flavor masking and may affect pectin gelation.

🔬 Thin-Film Oral Strips

The high lipid solubility and required therapeutic dosage of ligustilide often exceed the limited payload capacity of thin-film polymer matrices, leading to recrystallization or film brittleness.

For Brand Founders

Formulate with Angelica sinensis (Ligustilide)

Ready to launch a product featuring Angelica sinensis (Ligustilide)? Skip months of expensive wet-lab iterations. Generate a manufacturer-ready formulation in hours, instantly screened for physical incompatibilities and global regulatory compliance.

Build Science-Backed Formulation

Efficacy Evidence

Maximize Angelica sinensis (Ligustilide) Bioavailability

Need absolute proof that your Angelica sinensis (Ligustilide) extract actually absorbs? Stop blindly combining generic powders. Run a physics-based PBPK simulation to mathematically engineer peak clinical efficacy and targeted plasma concentrations.

Simulate Bioavailability

For R&D Labs & CDMOs

Angelica sinensis (Ligustilide) Degradation Testing

Is your Angelica sinensis (Ligustilide) payload degrading in the capsule before the expiration date? Stop waiting for costly bench testing. Run an accelerated digital twin to precisely model oxidation pathways and pH shifts before finalizing a manufacturing run.

Model Active Degradation