Home The Active Ingredient Matrix Celery Extract (Apigenin)

Formulation Intelligence

Celery Extract (Apigenin)

Accelerate your CDMO or DTC pipeline. Map the exact physiochemical constraints, bioavailability synergies, and optimal delivery mechanisms for Celery Extract (Apigenin).

Apigenin is a bioactive flavone that functions as a competitive antagonist of adenosine A1 receptors and a positive allosteric modulator of GABA-A receptors, providing potent anxiolytic and neuroprotective effects while inhibiting pro-inflammatory cytokines via the NF-κB pathway.

Verified Molecular Profiling (NIH PubChem)

PubChem CID

5280443

Molecular Weight

270.24 g/mol

XLogP3 (Lipophilicity)

1.7

IUPAC Name

5,7-dihydroxy-2-(4-hydroxyphenyl)chromen-4-one

Pharmacokinetic Synergies & Enhancers

Proven Synergy Pairings

  • L-Theanine for synergistic modulation of GABAergic pathways to enhance sleep quality
  • Magnesium Bisglycinate for potentiating neuromuscular relaxation and sedative efficacy

Biological Formulation Enhancers

  • Piperine for the inhibition of UDP-glucuronosyltransferase to prevent rapid first-pass metabolism
  • Lecithin for the formation of phytosomes to improve the intestinal permeability of the hydrophobic aglycone

Delivery System Constraints & Modeling

Every active compound behaves uniquely based on the physical matrix it is suspended in. Below are the known physical chemistry challenges for Celery Extract (Apigenin) across standard consumer modalities.

💊 Standard Capsules

The low bulk density of concentrated celery extract necessitates the use of high-flow lubricants like magnesium stearate to ensure consistent volumetric filling in high-speed encapsulation.

🍬 Gummy & Pectin Formats

Apigenin's hydrophobic nature and distinct herbal notes require complexation with cyclodextrins to prevent precipitation and maintain organoleptic neutrality in pectin-based matrices.

🔬 Thin-Film Oral Strips

The relatively high therapeutic threshold of apigenin poses a significant challenge for thin-film loading, often requiring micronization to maintain film integrity and rapid dissolution.

For Brand Founders

Formulate with Celery Extract (Apigenin)

Ready to launch a product featuring Celery Extract (Apigenin)? Skip months of expensive wet-lab iterations. Generate a manufacturer-ready formulation in hours, instantly screened for physical incompatibilities and global regulatory compliance.

Build Science-Backed Formulation

Efficacy Evidence

Maximize Celery Extract (Apigenin) Bioavailability

Need absolute proof that your Celery Extract (Apigenin) extract actually absorbs? Stop blindly combining generic powders. Run a physics-based PBPK simulation to mathematically engineer peak clinical efficacy and targeted plasma concentrations.

Simulate Bioavailability

For R&D Labs & CDMOs

Celery Extract (Apigenin) Degradation Testing

Is your Celery Extract (Apigenin) payload degrading in the capsule before the expiration date? Stop waiting for costly bench testing. Run an accelerated digital twin to precisely model oxidation pathways and pH shifts before finalizing a manufacturing run.

Model Active Degradation