Home The Active Ingredient Matrix Luteolin

Formulation Intelligence

Luteolin

Accelerate your CDMO or DTC pipeline. Map the exact physiochemical constraints, bioavailability synergies, and optimal delivery mechanisms for Luteolin.

Luteolin is a flavone that modulates neuroinflammation and cellular senescence by inhibiting the NF-κB and MAPK signaling pathways while activating Nrf2-mediated antioxidant defenses.

Verified Molecular Profiling (NIH PubChem)

PubChem CID

5280445

Molecular Weight

286.24 g/mol

XLogP3 (Lipophilicity)

1.4

IUPAC Name

2-(3,4-dihydroxyphenyl)-5,7-dihydroxychromen-4-one

Pharmacokinetic Synergies & Enhancers

Proven Synergy Pairings

  • Palmitoylethanolamide (PEA) for synergistic neuroprotective and anti-inflammatory effects in microglia
  • Quercetin for enhanced inhibition of mast cell degranulation and histamine release

Biological Formulation Enhancers

  • Piperine for inhibition of glucuronidation to increase systemic bioavailability
  • Lecithin for liposomal encapsulation to overcome poor aqueous solubility

Delivery System Constraints & Modeling

Every active compound behaves uniquely based on the physical matrix it is suspended in. Below are the known physical chemistry challenges for Luteolin across standard consumer modalities.

💊 Standard Capsules

Low bulk density and poor flowability of pure luteolin powder require specific excipients like microcrystalline cellulose to ensure uniform die filling.

🍬 Gummy & Pectin Formats

The intense yellow pigment of luteolin can cause significant staining of manufacturing equipment and may require high concentrations of masking agents to offset its inherent bitterness.

🔬 Thin-Film Oral Strips

The high dosage required for therapeutic efficacy often exceeds the 20-30mg payload capacity of standard polymer matrices in thin-film technology.

For Brand Founders

Formulate with Luteolin

Ready to launch a product featuring Luteolin? Skip months of expensive wet-lab iterations. Generate a manufacturer-ready formulation in hours, instantly screened for physical incompatibilities and global regulatory compliance.

Build Science-Backed Formulation

Efficacy Evidence

Maximize Luteolin Bioavailability

Need absolute proof that your Luteolin extract actually absorbs? Stop blindly combining generic powders. Run a physics-based PBPK simulation to mathematically engineer peak clinical efficacy and targeted plasma concentrations.

Simulate Bioavailability

For R&D Labs & CDMOs

Luteolin Degradation Testing

Is your Luteolin payload degrading in the capsule before the expiration date? Stop waiting for costly bench testing. Run an accelerated digital twin to precisely model oxidation pathways and pH shifts before finalizing a manufacturing run.

Model Active Degradation