Home The Active Ingredient Matrix Rutin

Formulation Intelligence

Rutin

Accelerate your CDMO or DTC pipeline. Map the exact physiochemical constraints, bioavailability synergies, and optimal delivery mechanisms for Rutin.

Rutin is a flavonol glycoside that exerts potent vasoprotective and antioxidant effects by inhibiting protein disulfide isomerase (PDI) and reducing capillary permeability.

Verified Molecular Profiling (NIH PubChem)

PubChem CID

5280805

Molecular Weight

610.5 g/mol

XLogP3 (Lipophilicity)

-1.3

IUPAC Name

2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-3-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-2-yl]oxychromen-4-one

Pharmacokinetic Synergies & Enhancers

Proven Synergy Pairings

  • Vitamin C for enhanced antioxidant regeneration and collagen synthesis support
  • Hesperidin for synergistic improvement of venous tone and microcirculation
  • Bromelain for enhanced anti-inflammatory response in soft tissue recovery

Biological Formulation Enhancers

  • Piperine for inhibition of glucuronidation to increase systemic bioavailability
  • Quercetin for potential metabolic sparing as they share similar aglycone pathways

Delivery System Constraints & Modeling

Every active compound behaves uniquely based on the physical matrix it is suspended in. Below are the known physical chemistry challenges for Rutin across standard consumer modalities.

💊 Standard Capsules

Rutin's low aqueous solubility necessitates micronization or the use of surfactants to ensure consistent dissolution rates within the gastrointestinal tract.

🍬 Gummy & Pectin Formats

The high dosage requirements for clinical efficacy often lead to significant texture degradation and a gritty mouthfeel in pectin-based matrices.

🔬 Thin-Film Oral Strips

Rutin's relatively high effective dose and hydrophobic nature make it difficult to load into thin-film polymers without compromising film flexibility and structural integrity.

For Brand Founders

Formulate with Rutin

Ready to launch a product featuring Rutin? Skip months of expensive wet-lab iterations. Generate a manufacturer-ready formulation in hours, instantly screened for physical incompatibilities and global regulatory compliance.

Build Science-Backed Formulation

Efficacy Evidence

Maximize Rutin Bioavailability

Need absolute proof that your Rutin extract actually absorbs? Stop blindly combining generic powders. Run a physics-based PBPK simulation to mathematically engineer peak clinical efficacy and targeted plasma concentrations.

Simulate Bioavailability

For R&D Labs & CDMOs

Rutin Degradation Testing

Is your Rutin payload degrading in the capsule before the expiration date? Stop waiting for costly bench testing. Run an accelerated digital twin to precisely model oxidation pathways and pH shifts before finalizing a manufacturing run.

Model Active Degradation