Home The Active Ingredient Matrix S-Adenosyl-L-Methionine (SAMe)

Formulation Intelligence

S-Adenosyl-L-Methionine (SAMe)

Accelerate your CDMO or DTC pipeline. Map the exact physiochemical constraints, bioavailability synergies, and optimal delivery mechanisms for S-Adenosyl-L-Methionine (SAMe).

SAMe serves as the primary methyl donor in the transmethylation cycle, critical for the synthesis of monoamine neurotransmitters, membrane phospholipids, and the maintenance of hepatic glutathione levels through the transsulfuration pathway.

Verified Molecular Profiling (NIH PubChem)

PubChem CID

34755

Molecular Weight

398.4 g/mol

XLogP3 (Lipophilicity)

-2.8

IUPAC Name

(2S)-2-amino-4-[[(2S,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-methylsulfonio]butanoate

Pharmacokinetic Synergies & Enhancers

Proven Synergy Pairings

  • Vitamin B12 for cofactor-dependent remethylation of homocysteine
  • 5-MTHF for sustaining the methionine cycle flux
  • Trimethylglycine for supporting the betaine-homocysteine methyltransferase pathway

Biological Formulation Enhancers

  • Enteric coating for protection against gastric acid-induced hydrolysis
  • Blister packaging for moisture exclusion to prevent hygroscopic degradation

Delivery System Constraints & Modeling

Every active compound behaves uniquely based on the physical matrix it is suspended in. Below are the known physical chemistry challenges for S-Adenosyl-L-Methionine (SAMe) across standard consumer modalities.

💊 Standard Capsules

Standard capsules require enteric coating to bypass gastric acidity and must be protected from moisture to prevent salt degradation.

🍬 Gummy & Pectin Formats

The high hygroscopicity and sensitivity to aqueous environments make SAMe highly unstable in gummy matrices, leading to rapid loss of biological activity.

🔬 Thin-Film Oral Strips

The high therapeutic dosage requirements of SAMe significantly exceed the physical loading capacity of thin-film oral delivery systems.

For Brand Founders

Formulate with S-Adenosyl-L-Methionine (SAMe)

Ready to launch a product featuring S-Adenosyl-L-Methionine (SAMe)? Skip months of expensive wet-lab iterations. Generate a manufacturer-ready formulation in hours, instantly screened for physical incompatibilities and global regulatory compliance.

Build Science-Backed Formulation

Efficacy Evidence

Maximize S-Adenosyl-L-Methionine (SAMe) Bioavailability

Need absolute proof that your S-Adenosyl-L-Methionine (SAMe) extract actually absorbs? Stop blindly combining generic powders. Run a physics-based PBPK simulation to mathematically engineer peak clinical efficacy and targeted plasma concentrations.

Simulate Bioavailability

For R&D Labs & CDMOs

S-Adenosyl-L-Methionine (SAMe) Degradation Testing

Is your S-Adenosyl-L-Methionine (SAMe) payload degrading in the capsule before the expiration date? Stop waiting for costly bench testing. Run an accelerated digital twin to precisely model oxidation pathways and pH shifts before finalizing a manufacturing run.

Model Active Degradation